Cilostazol 100 mg new

May 11, 2023

CILOSTAZONE 100 

Cilostazol 100

In the world of modern medicine, the management of vascular diseases and conditions related to poor blood circulation has become a key focus for medical practitioners. One drug that has gained considerable attention in this regard is Cilostazone 100, a medication primarily used to improve blood flow and reduce symptoms associated with peripheral arterial disease (PAD). With its active ingredient Cilostazol (100 mg), Cilostazone 100 plays a crucial role in enhancing circulation, improving exercise tolerance, and offering relief from intermittent claudication.

This article delves deep into the composition, benefits, key features, and usage of Cilostazone 100, explaining why it is an effective option for patients dealing with poor blood circulation and vascular problems. Additionally, a detailed FAQ section provides further insights into its usage, safety, and potential side effects.

Composition

Cilostazone 100 contains the active pharmaceutical ingredient Cilostazol (100mg). Cilostazol is a phosphodiesterase III inhibitor that works by dilating blood vessels and preventing blood clotting, thus improving circulation. It is an anti-platelet and vasodilator agent that also plays a role in inhibiting platelet aggregation, which can be critical in preventing clot formation in the arteries. This mechanism helps to alleviate the discomfort associated with poor circulation, particularly in conditions like peripheral arterial disease (PAD), where blood flow to the limbs is impaired.

Key Features and Ingredients

The core ingredient in Cilostazone 100 is Cilostazol, which serves as the cornerstone for its effectiveness. Below are some of the key features of Cilostazone 100 and its active ingredient, Cilostazol:

  1. Cilostazol (100 mg):

    • Mechanism of Action: Cilostazol works by inhibiting phosphodiesterase III (PDE3), which leads to increased cyclic AMP (cAMP) levels in platelets and blood vessel smooth muscle. This reduces platelet aggregation and promotes vasodilation (widening of blood vessels), leading to improved blood flow and reduced symptoms of claudication.
    • Vasodilation Effect: Cilostazol has the capacity to dilate blood vessels, thereby improving blood flow, particularly in the arteries of the legs, which is beneficial for individuals suffering from peripheral arterial disease (PAD).
    • Anti-Platelet Action: By reducing platelet aggregation, Cilostazol helps prevent the formation of blood clots, which could otherwise lead to more serious complications like stroke or heart attack.
  2. Other Excipients:

    • Cilostazone 100 may contain excipients such as starch, magnesium stearate, lactose, or microcrystalline cellulose. These inactive ingredients serve various purposes such as aiding in the drug's formulation, ensuring the tablet's stability, and improving the patient’s ability to swallow the pill.
  3. Tablet Formulation:

    • Cilostazone 100 is typically available as a tablet containing 100mg of Cilostazol, which makes it convenient for oral administration. The formulation ensures that patients can receive a precise dose of the active ingredient.

Usage

Cilostazone 100 is primarily used for the management of intermittent claudication, a condition where muscle pain occurs during exercise due to insufficient blood supply to the muscles. This condition is a hallmark symptom of peripheral arterial disease (PAD), a condition that occurs when the arteries in the legs become narrowed or blocked. The key indications for Cilostazone 100 include:

  1. Peripheral Arterial Disease (PAD):

    • Cilostazone 100 is prescribed to manage the symptoms of PAD. It helps improve walking distance and exercise tolerance in patients suffering from claudication, thereby enhancing their quality of life.
  2. Intermittent Claudication:

    • This condition, marked by pain in the leg muscles while walking or exercising, is the most common reason for prescribing Cilostazone 100. The medication helps alleviate this discomfort by improving blood flow and reducing ischemia (lack of oxygen due to poor circulation).
  3. Stroke Prevention:

    • Cilostazol, the active ingredient in Cilostazone 100, has been studied for its potential role in preventing strokes by inhibiting platelet aggregation and reducing the likelihood of clot formation.

Dosage and Administration:

  • The typical recommended dose of Cilostazone 100 is one tablet (100mg) taken twice daily, once in the morning and once in the evening, preferably after meals to minimize potential stomach irritation.
  • It is important to follow the prescribed dosage and not alter the dose without medical consultation, as overdose or misuse can lead to side effects.
  • Cilostazone 100 should not be used in combination with other medications that increase the risk of bleeding unless advised by a doctor.

Precautions:

  • Before starting Cilostazone 100, patients should inform their healthcare provider of any medical conditions, such as heart disease, liver dysfunction, or any history of bleeding disorders.
  • Pregnancy and Breastfeeding: Cilostazone 100 is generally not recommended during pregnancy or breastfeeding unless absolutely necessary. Women who are pregnant or planning to conceive should discuss potential risks with their healthcare provider.
  • Liver Function: Cilostazol should be used with caution in individuals with impaired liver function, as the drug is metabolized by the liver.

Benefits

Cilostazone 100 offers a wide array of benefits, particularly for patients dealing with vascular health issues. Some of the key benefits of Cilostazone 100 include:

  1. Improved Blood Flow:

    • The primary benefit of Cilostazone 100 is its ability to improve blood flow to the extremities, particularly in individuals with PAD. By widening blood vessels and improving circulation, the medication enhances oxygen delivery to tissues that are at risk of ischemia, thereby relieving symptoms like pain and cramping.
  2. Relieves Intermittent Claudication:

    • Cilostazone 100 is effective in reducing the symptoms of intermittent claudication, allowing patients to walk longer distances without experiencing discomfort. This significant improvement in mobility has a positive impact on overall quality of life.
  3. Prevention of Blood Clots:

    • Cilostazol inhibits platelet aggregation, helping prevent blood clots from forming in the arteries. This reduces the risk of serious cardiovascular events such as stroke, heart attack, or deep vein thrombosis (DVT).
  4. Improved Exercise Tolerance:

    • Patients taking Cilostazone 100 often experience improved exercise tolerance, meaning they can engage in physical activities without experiencing excessive fatigue or pain. This enhances overall physical fitness and well-being.
  5. Reduced Risk of Vascular Events:

    • By improving circulation and preventing clot formation, Cilostazone 100 can help reduce the risk of future vascular events, including heart attacks and strokes, which are particularly important for individuals with existing cardiovascular risk factors.
  6. Minimal Side Effects:

    • Cilostazone 100 is well-tolerated by many patients, and side effects are typically mild. Common side effects might include headaches or mild digestive discomfort, but serious adverse reactions are rare.

FAQ Section

Q1: How long does it take for Cilostazone 100 to show results?

  • It typically takes 2-4 weeks for patients to start noticing significant improvements in walking distance and reduced pain. However, the exact timeline can vary depending on individual health conditions and the severity of PAD.

Q2: Can I take Cilostazone 100 with other medications?

  • It is important to inform your doctor about all the medications you are currently taking, including over-the-counter drugs and supplements. Cilostazone 100 may interact with certain medications, particularly anticoagulants or antiplatelet drugs.

Q3: What should I do if I miss a dose of Cilostazone 100?

  • If you miss a dose of Cilostazone 100, take it as soon as you remember unless it is almost time for your next dose. In that case, skip the missed dose—do not double up to make up for a missed dose.

Q4: Is Cilostazone 100 safe for long-term use?

  • Cilostazone 100 is generally safe for long-term use, but regular monitoring by a healthcare provider is recommended to ensure continued effectiveness and safety, particularly in those with underlying health conditions.

Q5: Are there any dietary restrictions while taking Cilostazone 100?

  • There are no specific dietary restrictions associated with Cilostazone 100. However, it is advisable to maintain a healthy diet, avoid excessive alcohol, and follow any dietary recommendations provided by your healthcare provider.

Conclusion

In conclusion, Cilostazone 100 is an effective and reliable treatment option for individuals suffering from peripheral arterial disease, intermittent claudication, and related vascular issues. With its active ingredient Cilostazol, this medication improves blood flow, reduces pain, prevents blood clots, and enhances exercise tolerance. By incorporating Cilostazone 100 into a comprehensive treatment plan, patients can experience significant improvements in their quality of life, greater mobility, and a reduced risk of cardiovascular complications. 

About The Author

STERIS HEALTHCARE PVT LTD

Steris Healthcare Pvt Ltd, known as Sterispharma, was founded in February 2018 by a team of experienced professionals in the pharmaceutical industry. Headquartered in Navi Mumbai, the company holds certifications from WHO, GMP, and ISO, reflecting its dedication to maintaining high standards of quality and safety. Sterispharma’s mission is to provide affordable, high-quality medications across India, strictly adhering to WHO guidelines. With the convenience of an online pharmacy, customers can easily order medicines with home delivery options.

For further information 

Email: info@sterispharma.com / contact@sterispharma.com

Call/WhatsApp: 8209542042 , 8824175417

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